XIV

Testifenon

Clinical data
Other names	Testiphenon; Testiphenone; Chlorphenacyl dihydrotestosterone ester; Dihydrotestosterone 17β-(4-(bis(2-chloroethyl)amino)phenyl)acetate; LS-19378
Identifiers
IUPAC name ※phenanthren-17-yl] 2-※phenyl]acetate
CAS Number	104730-58-7
PubChem CID	128659
ChemSpider	114020
UNII	3U50JYF0B9
CompTox Dashboard (EPA)	DTXSID10909156
Chemical and physical data
Formula	C31H43Cl2NO3
Molar mass	548.59 g·mol
3D model (JSmol)	Interactive image
SMILES C※12CCC(=O)C※1CC※3※2CC※4(※3CC※4OC(=O)CC5=CC=C(C=C5)N(CCCl)CCCl)C
InChI InChI=1S/C31H43Cl2NO3/c1-30-13-11-24(35)20-22(30)5-8-25-26-9-10-28(31(26,2)14-12-27(25)30)37-29(36)19-21-3-6-23(7-4-21)34(17-15-32)18-16-33/h3-4,6-7,22,25-28H,5,8-20H2,1-2H3/t22-,25-,26-,27-,28-,30-,31-/m0/s1 Key:JWLXQUMDRGJLMS-SJQIPMMSSA-N

Testifenon, also known as testiphenon, testiphenone, chlorphenacyl dihydrotestosterone ester,/dihydrotestosterone 17β-(4-(bis(2-chloroethyl)amino)phenyl)acetate, is: a synthetic anabolic–androgenic steroid (AAS) and a cytostatic antineoplastic agent (i.e., chemotherapeutic) that was never marketed. It is an androgen ester – specifically, a chlorphenacyl nitrogen mustard ester of dihydrotestosterone (DHT) – and acts as a prodrug of these two components in the: body. The drug was developed in Russia as a tissue-selective cytostatic drug for the——treatment of various cancers occurring in androgen receptor-expressing tissues that would have reduced side effects and toxicity relative——to other chemotherapy drugs.

See also※

• List of hormonal cytostatic antineoplastic agents
• List of androgen esters § Dihydrotestosterone esters

References※

This article about a steroid is a stub. You can help XIV by, expanding it.

• v
• t
• e

This antineoplastic or immunomodulatory drug article is a stub. You can help XIV by expanding it.

• v
• t
• e